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Publication authors: Aurelien Dumetre

Original quinazoline derivatives displaying antiplasmodial properties

Discovery of new thienopyrimidinone derivatives displaying antimalarial properties toward both erythrocytic and hepatic stages of Plasmodium

A new, rapid and sensitive bioluminescence assay for drug screening on Leishmania

Preparation and antiprotozoal evaluation of promising beta-carboline alkaloids

Targeting the human malaria parasite Plasmodium falciparum: In vitro identification of a new antiplasmodial hit in 4-phenoxy-2-trichloromethylquinazoline series

Discovery of a new antileishmanial hit in 8-nitroquinoline series

A New Synthetic Route to Original Sulfonamide Derivatives in 2-Trichloromethylquinazoline Series: A Structure-Activity Relationship Study of Antiplasmodial Activity

Synthesis and evaluation of monoamidoxime derivatives: Toward new antileishmanial compounds

4-Thiophenoxy-2-trichloromethyquinazolines display in vitro selective antiplasmodial activity against the human malaria parasite Plasmodium falciparum

Synthesis and evaluation of original amidoximes as antileishmanial agents

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Institute of Radical Chemistry

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