Skip to content
  • Intranet
  • Annuaire
  • Contact
Menu
  • Intranet
  • Annuaire
  • Contact
Search
  • Institut
    • Annuaire
    • Contact
    • Groupe de travail
    • Présentation
  • Équipes
    • Chimie Moléculaire Organique
    • Chimie Radicalaire Appliquée à la Biologie
    • Chimie Radicalaire Organique et Polymères de Spécialité
    • Chimie Théorique
    • Pharmaco-Chimie Radicalaire
    • Sondes Moléculaires en Biologie et Stress Oxydant
    • Spectrométries Appliquées à la Caractérisation Structurale
    • Structure et Réactivité des Espèces Paramagnétiques
  • Publications
    • Articles
      • 2009
      • 2010
      • 2011
      • 2012
      • 2013
      • 2014
      • 2015
      • 2016
      • 2017
      • 2018
      • 2019
      • 2020
      • 2021
      • 2022
    • Brevets
  • News
  • Événement
  • Plateforme
    • Analyse polymère
    • Service Commun de RPE
  • Recrutement
Menu
  • Institut
    • Annuaire
    • Contact
    • Groupe de travail
    • Présentation
  • Équipes
    • Chimie Moléculaire Organique
    • Chimie Radicalaire Appliquée à la Biologie
    • Chimie Radicalaire Organique et Polymères de Spécialité
    • Chimie Théorique
    • Pharmaco-Chimie Radicalaire
    • Sondes Moléculaires en Biologie et Stress Oxydant
    • Spectrométries Appliquées à la Caractérisation Structurale
    • Structure et Réactivité des Espèces Paramagnétiques
  • Publications
    • Articles
      • 2009
      • 2010
      • 2011
      • 2012
      • 2013
      • 2014
      • 2015
      • 2016
      • 2017
      • 2018
      • 2019
      • 2020
      • 2021
      • 2022
    • Brevets
  • News
  • Événement
  • Plateforme
    • Analyse polymère
    • Service Commun de RPE
  • Recrutement

Publication authors: Pierre Verhaeghe

Original quinazoline derivatives displaying antiplasmodial properties

Determination of uremic solutes in biological fluids of chronic kidney disease patients by HPLC assay

Tandem synthesis and in vitro antiplasmodial evaluation of new naphtho[2,1-d] thiazole derivatives

Looking for new antileishmanial derivatives in 8-nitroquinolin-2(1H)-one series

Discovery of new thienopyrimidinone derivatives displaying antimalarial properties toward both erythrocytic and hepatic stages of Plasmodium

Antileishmanial pharmacomodulation in 8-nitroquinolin-2(1H)-one series

Using the Sonogashira Reaction for Preparing a New Fragment Library based on the 3-alkynylimidazo[1,2-alpha] pyridine Scaffold

Discovery of new hit-molecules targeting Plasmodium falciparum through a global SAR study of the 4-substituted-2-trichloromethylquinazoline antiplasmodial scaffold

Synthesis of antiplasmodial 2-aminothieno[3,2-d]pyrimidin-4(3H)-one analogues using the scaffold hopping strategy

A new, rapid and sensitive bioluminescence assay for drug screening on Leishmania

A new DMAP-catalyzed and microwave-assisted approach for introducing heteroarylamino substituents at position-4 of the quinazoline ring

Synthesis and in vitro evaluation of 4-trichloromethylpyrrolo[1,2-a]quinoxalines as new antiplasmodial agents

Targeting the human parasite Leishmania donovani: Discovery of a new promising anti-infectious pharmacophore in 3-nitroimidazo[1,2-a]pyridine series

Sonogashira cross-coupling reaction in 4-chloro-2-trichloromethylquinazoline series is possible despite a side dimerization reaction

Safety Review: Squalene and Thimerosal in Vaccines

Targeting the human malaria parasite Plasmodium falciparum: In vitro identification of a new antiplasmodial hit in 4-phenoxy-2-trichloromethylquinazoline series

Discovery of a new antileishmanial hit in 8-nitroquinoline series

A New Synthetic Route to Original Sulfonamide Derivatives in 2-Trichloromethylquinazoline Series: A Structure-Activity Relationship Study of Antiplasmodial Activity

Synthesis and evaluation of monoamidoxime derivatives: Toward new antileishmanial compounds

First SNAr reaction using TDAE-initiated carbanions in quinazoline series

4-Thiophenoxy-2-trichloromethyquinazolines display in vitro selective antiplasmodial activity against the human malaria parasite Plasmodium falciparum

Regioselective Suzuki-Miyaura Reaction: Application to the Microwave-promoted Synthesis of 4,7-Diarylquinazolines

Access to Original Vinylic Chlorides in the Quinazoline Series via a Monoelectronic Transfer Reaction Approach

Looking for new antiplasmodial quinazolines: DMAP-catalyzed synthesis of 4-benzyloxy- and 4-aryloxy-2-trichloromethylquinazolines and their in vitro evaluation toward Plasmodium falciparum

Synthesis and Antiplasmodial Evaluation of 4-Carboxamido- and 4-Alkoxy-2-Trichloromethyl Quinazolines

2-Phenoxy-3-Trichloromethylquinoxalines Are Antiplasmodial Derivatives with Activity against the Apicoplast of Plasmodium falciparum

Antikinetoplastid SAR study in 3-nitroimidazopyridine series: Identification of a novel non-genotoxic and potent anti-T.b. brucei hitcompound with improved pharmacokinetic properties

8-Alkynyl-3-nitroimidazopyridines display potent antitrypanosomal activity against both T. b. brucei and cruzi

Anticancer and Anti-Inflammatory Activities of Some New Pyrazolo[3,4-b]pyrazines

8-Aryl-6-chloro-3-nitro-2-(phenylsulfonylmethyl)imidazo[1,2-a] pyridines as potent antitrypanosomatid molecules bioactivated by type 1 nitroreductases

Nongenotoxic 3-Nitroimidazo[1,2-a]pyridines Are NTR1 Substrates That Display Potent in Vitro Antileishmanial Activity

  • Intranet
  • Annuaire
  • Contact
  • Mentions Légales
Menu
  • Intranet
  • Annuaire
  • Contact
  • Mentions Légales

Welcome to

Institute of Radical Chemistry

Lost your password?
blank
blank
blank